Vanadium-catalyzed asymmetric oxidation of alpha-hydroxy esters using molecular oxygen as stoichiometric oxidant.

نویسندگان

  • Alexander T Radosevich
  • Christine Musich
  • F Dean Toste
چکیده

A vanadium-catalyzed method for the oxidative kinetic resolution of alpha-hydroxyesters, using oxygen as the terminal oxidant, is described. The catalyst is generated in situ from vanadium(V) tri-iso-propoxyoxide in combination with a tridentate ligand derived from 3,5-di-tert-butylsalicylaldehyde and (S)-tert-leucinol. The reaction allows for the enantioselective synthesis of both aromatic and aliphatic secondary alcohols, including those containing olefins and alkynes.

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عنوان ژورنال:
  • Journal of the American Chemical Society

دوره 127 4  شماره 

صفحات  -

تاریخ انتشار 2005